Selective Immunoproteasome Inhibition

Selective Immunoproteasome Inhibition

Title
DiscoveryDisc
Phase 1Ph1
Phase 2Ph2
Phase 3Ph3

Zetomipzomib (KZR-616)

Lupus Nephritis (LN)

Zetomipzomib (KZR-616)

Lupus Nephritis (LN)
PALIZADEPALIZADE
Autoimmune Hepatitis (AIH)
Autoimmune Hepatitis (AIH)
PORTOLAPORTOLA
Dermatomyositis (DM) Polymyositis (PM)
Dermatomyositis (DM) Polymyositis (PM)
PRESIDIO OLEPRESIDIO OLE

Protein Secretion Inhibition

Protein Secretion Inhibition

Title
DiscoveryDisc
Phase 1Ph1
Phase 2Ph2
Phase 3Ph3

KZR-261

Advanced/Metastatic Solid Tumor

KZR-261

Advanced/Metastatic Solid Tumor

Oral Anti-PD-1

Single Target Oncology

Oral Anti-PD-1

Single Target Oncology

KZR-TBD

Multi Target Oncology

KZR-TBD

Multi Target Oncology